Percentage of Excipients Used in Tablet Formulation


Pharmaceutical Tablets are solid dosage forms containing drug substances usually prepared with the aid of suitable pharmaceutical excipients. Here we mention a list of common pharmaceutical excipients used in tablet formulation.


A List of Excipients Used in Tablet Formulation

Alginic Acid -  1 to 5% w/w (as both a binder and disintegrating agent)

Alpha Tocopherol - 0.001 to 0.05% v/v (as an antioxidant for oil- or fat-based product)

Aspartame – 180 to 200 times more sweetener than sucrose

Butylated Hydroxyanisole – 0.01% (as an antioxidant)

Butylated hydroxytoluene - 0.01 to 0.1% (as an antioxidant)

Calcium Carbonate – amount may vary (as a diluent or bulking agent)

Dibasic Calcium Phosphate - amount may vary (to improve compaction properties or flow properties)

Calcium Stearate – up to 1.0% (as a lubricant)

Carbomer – 0.75 to 3% (as a binder)

Carbomer – 5 to 30% (as a control releasing agent)

Carboxymethylcellulose Sodium - 1 to 6% (as a binder)

Cellulose acetate phthalate (CAP) – 0.5 to 9% (as a coating agent)

Croscarmellose Sodium – up to 5% (as a disintegrant)

Crospovidone – 2 to 5% (as a disintegrant)

Hydroxypropyl cellulose – 2 to 6% (as a binder)

Hydroxypropyl cellulose – 15 to 35% (as an extended release polymer)

Hydroxypropyl Cellulose, Low-substituted – 5 to 50% (as a binder or disintegrant)

Hypromellose (HPMC) - 2 to 5% (as a binder)

Hypromellose (HPMC) – 10 to 80% % (as matrix forming agent)

Lactose, Monohydrate - amount may vary (as a diluent)

Lactose, Spray-Dried - amount may vary (as a diluent for moisture sensitive product)

Magnesium Stearate – 0.25 to 5% (as a lubricant)

Mannitol – 10 to 90% (as a diluent)

Microcrystalline cellulose – 20 to 90% (as a diluent)

Microcrystalline cellulose – 5 to 15% (as a disintegrant)

Poloxamer – 0.01 to 5% (as wetting agent)

Povidone – 0.5 to 5% (as a binder)

Pregelatinized starch – 5 to 75% (as a diluent)

Pregelatinized starch – 5 to 20% (as a binder)

Pregelatinized starch – 5 to 10% (as a disintegrant)

Saccharin – 0.02 to 0.5% (as a sweetening agent)

Silicified Microcrystalline cellulose - amount may vary (as a filler)

Stearic Acid – 1 to 3% (as a lubricant)

Talc – 1 to 10% (as a glidant and lubricant)

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